Unsaturated carboxylic acids in the one-pot synthesis of novel derivatives of 3,4-dihydro-2H-thiopyran reagent with maleic, itaconic, or 5-norbornene-2,3-dicarboxylic acid led to the corresponding
3,4-dihydro
Azidothymidine "clicked" into 1,2,3-Triazoles: First Report on Carbonic Anhydrase-Telomerase Dual-Hybrid InhibitorsBerrino E.,
Angeli A.,
Zhdanov D.D.,
Kiryukhina A.P.,
Milaneschi A.,
Bozdag M.,
Carradori S.,
Selleri S.,
Bartolucci G.,
Peat T.S.,
Ferraroni M.,
Supuran C.T.,
Carta F.,
De Luca A. from 5.2 to 9.1 μM). High-resolution X-ray crystallography on selected derivatives in the adduct with
h Intramolecular cascade annulation triggered by rhodium(III)catalyzed sequential C(sp 2 )–H activation and C(sp 3 )–H amination-hydroxyacrylamides for the construction of indolizinones via sequential C(sp 2 )–
H activation and C(sp 3 )–
H amination has been developed