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Benzothiazinones Kill Mycobacterium tuberculosis by blocking Arabinan synthesis

Дата публикации: 2021-04-27

Дата публикации в реестре: 2021-10-05T18:23:41Z

Аннотация:
Ключевые слова:
1,3 benzothiazinon 4 one, 2 [2 methyl 1,4 dioxa 8 azaspiro[4.5]dec 8 yl] 8 nitro 6 (trifluoromethyl) 4h 1,3 benzothiazin 4 one, arabinan, arabinose, bacterial enzyme, btz 038, btz 043, btz 044, decaprenylphosphoryl arabinose, decaprenylphosphoryl beta dextro ribose 2' epimerase, ethambutol, green fluorescent protein, isoniazid, tuberculostatic agent, unclassified drug, 2 (2 methyl 1,4 dioxa 8 azaspiro(4.5)dec 8 yl) 8 nitro 6 (trifluoromethyl) 4H 1,3 benzothiazin 4 one, 2-(2-methyl-1,4-dioxa-8-azaspiro(4.5)dec-8-yl)-8-nitro-6-(trifluoromethyl)-4H-1,3-benzothiazin-4-one, araban, decaprenylphosphoryl beta D ribose 2' epimerase, mouse, decaprenylphosphoryl-beta-D-ribose 2'-epimerase, mouse, enzyme inhibitor, ethambutol, isomerase, polysaccharide, spiro compound, thiazine derivative, tuberculostatic agent, bacterium, biochemistry, cell organelle, drug, genetic analysis, lysis, tuberculosis, animal experiment, animal model, antibacterial activity, article, bactericidal activity, chronic disease, controlled study, drug efficacy, drug potency, drug screening, drug structure, drug synthesis, drug targeting, enzyme inhibition, fluorescence microscopy, minimum inhibitory concentration, mouse, multidrug resistance, Mycobacterium, Mycobacterium tuberculosis, nonhuman, priority journal, structure activity relation, toxicity testing, treatment outcome, tuberculosis, amino acid sequence, animal, antibiotic resistance, bacterial gene, Bagg albino mouse, biosynthesis, cell wall, cerebrospinal fluid, chemical structure, chemistry, drug antagonism, drug effect, gene expression regulation, genetics, metabolism, microbiological examination, microbiology, molecular genetics, synthesis, tuberculosis, Bacteria (microorganisms), Mycobacterium tuberculosis, Amino Acid Sequence, Animals, Antitubercular Agents, Arabinose, Cell Wall, Drug Resistance, Bacterial, Enzyme Inhibitors, Ethambutol, Gene Expression Regulation, Bacterial, Genes, Bacterial, Mice, Mice, Inbred BALB C, Microbial Sensitivity Tests, Molecular Sequence Data, Molecular Structure, Mycobacterium, Mycobacterium tuberculosis, Polysaccharides, Racemases and Epimerases, Spiro Compounds, Thiazines, Tuberculosis

Тип: info:eu-repo/semantics/journal-article


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